Enzyme Modulators

Enzyme modulators are chemical compounds able to inhibit or activate enzymes. This product category includes modulators of various enzyme classes, such as oxidoreductases, transferases, hydrolases, lyases, isomerases and ligases. We offer a rich collection of kinase inhibitors and other enzymes involved in cell signalling, which are key tools for cancer research, cell biology, physiology and others.

产品编码 CAS号 产品名称 描述
BA166127 1384424-80-9

A 1070722

GSK-3α and GSK-3β inhibitor; reduces phosphorylation of Tau protein
FA17735 78957-85-4

A 3

Inhibitor of PKA kinase
BA166476 1889279-16-6

A 485

Histone acetyltransferase inhibitor of p300/CBP; anti-proliferative
BA41291 1166227-08-2

A 66 NEW

Inhibitor of PI3K kinase; anti-cancer agent; arrhythmogenic
FA16147 844499-71-4

A 769662

Activates AMP-activated protein kinase (AMPK)
BA162484 909910-43-6

A 83-01

Inhibitor of TGF-β type I receptor ALK5 kinase
FA64929 959122-11-3

A 922500

DGAT-1 enzyme antagonist
BA162794 1032229-33-6

A 939572

Inhibitor of stearoyl-CoA desaturase 1
BA166584 1037826-77-9

A 953227

Calpain antagonist
FA100934 934162-61-5

A 966492

Inhibitor of PARP enzyme
BA164085 1982372-88-2


Inhibitor of histone-lysine N-methyltransferase SUV420H1 and SUV420H2
FE103812 1231929-97-7


Inhibitor of cyclin-dependent kinases CDK4 and CDK6
FA159696 1231930-82-7

Abemaciclib mesylate

Inhibits cyclin-dependent kinase 4 and 6 (CDK4 and CDK6); antineoplastic
BA164060 154229-19-3


CYP17 enzyme inhibitor
BA164133 154229-18-2

Abiraterone acetate

CYP17 enzyme inhibitor

Abiraterone ethyl ether

CYP17 enzyme inhibitor
FA166721 1310726-60-3

ABT 494

Inhibitor of Janus kinase JAK-1
FF100506 154355-76-7

ABT 761

Inhibitor of 5-lipoxygenase
FA138815 1420477-60-6


Inhibitor of the Bruton tyrosine kinase
FA101029 870281-34-8


 Selective PI3Kδ inhibitor
BA164135 89796-99-6


Cyclooxygenase inhibitor; NSAID
FA16912 53164-05-9


Non-steroidal anti-inflammatory drug
FA17211 18699-02-0


Inhibitor of IL-1 secretion; anti-inflammatory; immunomodulatory
BA164806 1316214-52-4

ACY 1215

Inhibitor of histone deacetylase 6
BA164139 142340-99-6

Adefovir dipivoxil

Anti-viral; reverse transcriptase inhibitor
FA17224 791828-58-5


Dual inhibitor of ADAM10 and ADAM17 metalloproteases
FA17229 497839-62-0

AEE 788

Dual inhibitor of EGFR and VEGR receptor phosphorylation; anti-metastatic
BA164141 850140-72-6


Irreversible inhibitor of ErbB1, ErbB2/HER2 and ErbB4 receptor tyrosine kinases
FA103643 439081-17-1


Irreversible inhibitor of ErbB1, ErbB2/HER2 and ErbB4; less active enantiomer
BA162012 850140-73-7

Afatinib dimaleate

Irreversible inhibitor of ErbB1, ErbB2/HER2 and ErbB4 receptor tyrosine kinases
BA166066 1047644-62-1


Inhibitor of pan-AKT
FA145491 1448347-49-6


Inhibits mutant form of IDH-1 enzyme; anti-proliferative
FA145490 1446502-11-9

AG 221

Inhibitor of isocitrate dehydrogenase 2
FC17241 134036-52-5

AG 490

Inhibits EGFR, STAT3, JAK3/STAT, JAK3/AP-1 and JAK3/MAPK tyrosine kinases
BA166653 681281-88-9

Akt Inhibitor IV

Inhibitor of Akt kinase
FA17261 1483-07-4


Inhibitor of glutaminase; glutamine analogue
FA64934 1256589-74-8

Alectinib HCl

Active product of vitamin A metabolism
BA164144 121268-17-5

Alendronic acid monosodium salt trihydrate

Farnesyl diphosphate synthase inhibitor; inhibits bone resorption
BA165582 1245916-14-6


Monoclonal antibody to PCSK9 ; inhibitor of proprotein convertase PCSK9
BA164146 173334-58-2

Aliskiren hemifumarate

Non-peptide renin inhibitor; anti-hypertensive
FA17288 315-30-0

Allopurinol - EP grade

Inhibitor of xanthine oxidase and urate synthesis
FA137645 1345847-93-9


Inhibitor of MET, TIE2 and VEGFR2 kinases
BA164807 1186206-79-0


Eph receptor tyrosine kinase inhibitor
BA166478 179044-97-4

AMG 18 hydrochloride

Inhibitor of endonuclease IRE1α
FA64937 913376-83-7

AMG 458

c-Met receptor tyrosine kinase inhibitor
FA137647 1401033-86-0

AMG 925

Dual inhibitor of FLT3 and CDK4 kinases
FA17375 385769-84-6

Amino tadalafil

Tadalafil analogue; PDE 5 inhibitor
BA164155 125-84-8


Aromatase inhibitor; anti-neoplastic
BA166016 317-34-0


Phosphodiesterase inhibitor
BA164161 68302-57-8


Inhibits serine/threonine-protein kinase TBK1 and IKKε enzyme; anti-allergic
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