Ion Channels

Ion channels are transmembrane proteins with the ability to control ion currents across cell membrane. They are essential for maintaining resting membrane potential as well as for generation of action potentials in neurons, muscle and endocrine cells. Our collection of ion channel modulators include blockers of ligand-gated and voltage-gated channels, as well as mechanosensitive, cyclic nucleotide-gated channels and more.

产品编码 CAS号 产品名称 描述
BE166951 945828-50-2

AA 29504

Allosteric GABAA receptor modulator; anxiolytic
BA164134 77337-73-6

Acamprosate calcium

GABA receptor agonist; threatment for alcohol dependence
BA165790 865305-30-2

AF 353

Antagonist of P2X3/P2X2/3 purinoreceptors

Ambroxol HCl

Antioxidant; secretolytic; anti-inflammatory; sodium channel blocker
FA164880 545395-94-6

AMG 9810

Vanilloid receptor 1 antagonist
FA61531 17440-83-4

Amiloride hydrochloride

Sodium channel inhibitor; inhibitor of urokinase-type plasminogen activator
BA139263 1951-25-3

Amiodarone hydrochloride

Multi-channel blocker; anti-arrhythmic agent
BA164164 88150-42-9

Amlodipine base

Inhibits L-type calcium channels; anti-hypertensive; antianginal
BA164162 111470-99-6

Amlodipine besylate

Inhibits L-type calcium channels; anti-hypertensive; antianginal
BA164165 88150-47-4

Amlodipine maleate

Inhibits L-type calcium channels; anti-hypertensive; antianginal
BA165665 926023-82-7


TRPM8 channel blocker
FA17896 3471-05-4


Natural neurotoxin
BA164183 72432-10-1


AMPA/kainate desensitization inhibitor
BA167283 2196197-89-2

AP 202

α4β2 nAChR antagonist; reduces nicotine self-administration in vivo
FA145501 178419-42-6

AR-R 17779 hydrochloride

Agonist of α7 nicotinic receptor
FA52437 14923-17-2

Arcaine Sulfate

Antagonist of NMDA receptor
FA18027 64228-81-5

Atracurium besylate

Nicotinic AChR antagonist; neuromuscular blocking agent; muscle relaxant
FA18062 123040-69-7

Azasetron hydrochloride

Serotonin 5-HT3 receptor antagonist; anti-emetic
FA158515 345303-91-5

AZD 9056 hydrochloride

P2X7 receptor antagonist
FB18144 104757-53-1

Barnidipine hydrochloride

Calcium channel blocker
BB162780 71145-03-4

BAY K 8644

Activates L-type Ca2+ channels; vasoconstrictive
BB165272 393514-24-4


Antagonist of vanilloid receptor TRPV1 
FB64953 91599-74-5

Benidipine hydrochloride

Calcium channel blocker 
BB164251 485-49-4


Inhibitor of ionotropic receptor GABA(A)
BB162664 40709-69-1

(-)-Bicuculline methiodide

Inhibitor of ionotropic receptor GABA(A); less active isomer
FB157252 11032-79-4


Antagonist of nicotinic acetylcholine receptors; neurotoxin
BB166160 2180-92-9


Sodium channel blocker, targets channel intracellular domain
BC166161 298-46-4


GABA agonist; voltage-gated sodium channel blocker
FC19680 36507-30-9

Carbamazepine 10,11-epoxide

Inhibitor of neuronal voltage-gated sodium channels
FC158497 724424-43-5

CE 224,535

Antagonist of purinoreceptor P2X7
BC164309 132203-70-4


Inhibits L- and N-type calcium channels; anti-hypertensive; neuroprotective
BC167081 298-57-7


Calcium channel blocker; piperazine derivative
FC74963 92953-10-1

Clofilium tosylate

Potassium channel blocker; anti-arrhythmic; cardiac depressant
FC20628 115066-14-3


Glutamate antagonist
FC20595 215923-54-9

CX 546

AMPA receptor potentiator
BC164343 485-35-8


Nicotinic ACh receptor agonist
BD162474 79055-68-8


Antagonist of NMDA receptor
BD162627 29734-68-7

Dihydro-b-erythroidine hydrobromide

Antagonist of nicotinic receptor
BD166408 33286-22-5


L-type calcium channel blocker
BD162539 76326-31-3


Antagonist of NMDA receptor
FD22437 2379-57-9


AMPA/ kainate receptor antagonist 
BD164377 115256-11-6


Potassium channel blocker; antiarrhythmic agent
FD14809 115956-13-3

Dolasetron mesylate

Serotonin receptor 5-HT3 antagonist
FD61522 113-07-5

Doxapram hydrochloride

Inhibitor of TASK tandem pore potassium channel; respiratory stimulant
BD164395 141625-93-6

Dronedarone hydrochloride

Multichannel blocker; reduces sodium and calcium currents
FE162097 1262780-97-1


Agonist of calcium sensing receptor CASR; calcimimetic agent
FF23236 119945-59-4


Voltage-gated calcium channel blocker
BF164445 72509-76-3


L-type calcium channel blocker; anti-hypertensive
BF160700 78538-74-6

FG 7142

Agonist of benzodiazepine receptor; anxiogenic
FF23323 530-78-9

Flufenamic acid 氟灭酸

Inhibitor of calcium-activated non-selective cation channels
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